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Publications from CBMR

30. Autocatalytic and DMSO-Promoted Regioselective Synthesis of Pyrimidine-Fused Quinolines from Anilines and Barbituric Acids; 

 

 

 

 

 

 

 

P Yadav, D Chatterjee, S Bhowmick, K Tiwari, A Awasthi, Dharmendra Kumar Tiwari* Chemical Communications​​; 2024, (https://doi.org/10.1039/D4CC04044A)

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 29. Tf2O-mediated [4+2]-annulation of anthranils with 2-chloropyridines: enabling access to  pyrido-quinazolinones and euxylophoricine B; 

 

 

 

 

A. Awasthi,   K. Tiwari, and Dharmendra Kumar Tiwari* Chemical Communications​​; 202460, 7749 - 7752.

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28. Synthesis of 4-styrylquinolines via direct oxidative C3-alkenylation of anthranils under Pd(ii) catalysis:

 

 

 

 

 

 

 

A. Awasthi,   K. Tiwari,   P. Yadav,   S. Bhowmick and  Dharmendra Kumar Tiwari*; Chemical Communications​​; 20242054-2057

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27. DMSO as a dual carbon synthon in the one-pot tandem synthesis of N-alkylated quinazolinone from anthranilamides and acetophenones. P. Yadav,  S. Yadav,   A.  Awasthi,   M. Phanindrudu,   S. Bhowmick,   and  Dharmendra Kumar Tiwari*, New J. Chem., 2022, 46, 16289-16296

26. Copper-Catalyzed Synthesis of 3-Nitro-Quinolines from Nitro-Olefins and Anthranils: Its Application in the Synthesis of Quindoline; A.  Awasthi, P.  Yadav,  S.  Yadav,  and Dharmendra Kumar Tiwari,*  Advanced Synthesis & Catalysis,  2022, 364, 41 - 46

25. Stereoselective synthesis of (Z)-1,3-bis(α,β-unsaturated carbonyl)-isoindolines from aldehydes and phenacyl azides under metal-free conditions; B. Prasad, M. Phanindrudu,  J. B.  Nanubolu, A. Kamal, and Dharmendra Kumar Tiwari* Chem. Commun.,  2021, 57, 9542 - 9545. 

24. DMSO as a Methine Source in TFA-Mediated One-Pot Tandem Regioselective Synthesis of 3-Substituted-1-Aryl-1H-Pyrazolo-[3,4-b]quinolines from Anilines and Pyrazolones. P. Yadav, A. Awasthi, S. Gokulnath and Dharmendra Kumar Tiwari* J. Org. Chem. 2021, 86, 2658–2666.

23. A three-component, general and practical route for diastereoselective synthesis of aza-spirocyclic pyrazolones via a decarboxylative annulation process. A. Awasthi,  P. Yadav, and  Dharmendra Kumar Tiwari* New Journal of Chemistry, 2021, 45, 2374-2383.

22. α-Amino Acids Mediated C–C Double Bonds Cleavage in Diastereoselective Synthesis of Aza‐Spirocyclic Pyrazolones. A. Awasthi, P. Yadav; V.  Kumar; Dharmendra Kumar Tiwari* Advanced Synthesis & Catalysis, 2020, 362, 4378 - 4383.

21. Nano copper-catalyzed synthesis of symmetrical/unsymmetrical sulfones from aryl/alkyl halides and p-toluenesulfonyl-methylisocyanide: TosMIC as a tosyl source. M. Phanindrudu P. Jaya, P. R. Likhar, Dharmendra Kumar Tiwari*, Tetrahedron, 2020, 76, 131263.

 

20. Transition Metal-Free One-Pot Tandem Synthesis of 3-Ketoisoquinolines from Aldehydes and Phenacyl azides; B. Prasad, M. Phanindrudu, Dharmendra Kumar Tiwari* and A. Kamal; J. Org. Chem. 2019, 84, 12334–12343.

19. Synthesis of 3-keto-quinolines from enaminones, anilines, and DMSO: Transition metal-free one-pot cascade: S. B. Wakade, D. K. Tiwari, M. Phanindrudu, P. Yadav,  and Dharmendra Kumar Tiwari* , Tetrahedron, 2019, 75, 4024-4030.

18. A multicomponent reaction for the synthesis of pyrido [1,2-b] isoquinoline derivatives via the [3+2] cycloaddition reaction between alkynes and in situ generated isoquinolinium ylides; S.  S. Shinde,  S. Laha, Dharmendra K. Tiwari, B. Sridhar  and  Pravin R. Likhar; Org. Biomol. Chem., 2019, 17,  4121-412.

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Publications from DST-INSPIRE Faculty

17. Transition Metal-Free Approach for the Syntheses of 4-Aryl-quinolines from Alkynes and Anilines; M. PhanindruduS. B. WakadeDipak Kumar TiwariPravin R. Likhar, and Dharmendra Kumar Tiwari*; J. Org. Chem. 2018, 83, 9137–9143.

16. Transition Metal-Free Quinoline Synthesis from Acetophenones and Anthranils via Sequential One Carbon Homologation/Conjugate addition/Annulation Cascade: S. B. Wakade, D. K. Tiwari, P. S. K. P. Ganesh, M. Phanindrudu, P. Likhar, and Dharmendra Kumar Tiwari*; Organic Letters, 2017; 19, 4948.

15. α,β-Functionalization of Saturated Ketones with Anthranils via Cu-catalyzed Sequential Dehydrogenation/Aza-Michael Addition/Annulation Cascade Reactions in One-Pot: D. K. Tiwari, M. Phanindrudu, J. B. Nanubolu, and Dharmendra Kumar Tiwari*Chemical Communications,  2017, 53, 5302.

14. Unprecedented Synthesis of 1,2,3-Triazolo-Cinnolinone via Sonogashira Coupling and Intramolecular Cyclization; Avnish Kumar, Dharmendra Kumar Tiwari, Balasubramanian Sridhar, and Pravin R. Likhar; Org. Biomol. Chem., 2018,16, 4840-4848.

13. Magnetically Separable Nano Copper-Catalyzed Unprecedented Stereoselective Synthesis of E-Vinyl Sulfones from Tosylmethyl isocyanide and alkynes: TosMIC as a Source of Sulfonyl group; M. Phanindrudu, D. K. Tiwari, B. Sridhar, P. R. Likhar, and Dharmendra Kumar Tiwari*; Org. Chem.  Frontiers 2016; 3, 795 (Selected for Front Cover Image).

12. Magnetically Recoverable Cu0/Fe3O4 Catalyzed One-Pot Tandem Synthesis of Sulfur-Containing Triazoles from Alkynes and Azide: DMSO acts as an alkylating agent. M. Phanindrudu, Dipak Kumar Tiwari, V. K. Aravilli, K. C. Bhardwaj, G. Sabapathi, Pravin R. Likhar, and Dharmendra Kumar Tiwari,* Eur. J. Org. Chem. 2016, 4629.

11. Magnetically Recoverable Cu0/Fe3O4 Catalyzed Highly Regioselective Synthesis of 2,3,4-Trisubstituted Pyrroles     From Unactivated Terminal Alkynes and Isocyanides; D. K. Tiwari, M. Phanindrudu, V. K. Aravilli, B. Sridhar, Pravin R. Likhar and Dharmendra Kumar Tiwari*; Chemical Communications.; 2016, 52, 4675

​ 10. Palladium Catalyzed Domino Reaction of 1,4-Disubstituted 1,2,3-Triazoles via Double C-H functionalization: One-pot Synthesis of Triazolo[1,5-f]phenanthridines; Avanish Kumar, Dharmendra Kumar Tiwari, and Pravin Likhar; RSC Advances 2016, 6, 43638.

 9. Visible Light Photoredox Mediated sp3C-H Functionalization and Coupling of Secondary Amines with Vinyl Azides in Flow Microreactors; Dharmendra Kumar Tiwari,* R. Maurya* and J. B. Nanubolu; Chemistry-A European Journal, 2016, 22, 526.

 8. Nano-copper catalysed highly regioselective synthesis of 2,4-disubstituted pyrroles from terminal alkynes and isocyanides. D. K. Tiwari, J. Pogula, Dharmendra Kumar Tiwari* and Pravin R. Likhar, Chemical. Communications. 2015, 51, 13646

 7. A general and practical route to 4,5-disubstituted oxazoles using acid chlorides and isocyanides. Dipak Kumar Tiwari, Jaya Pogula, Dharmendra Kumar Tiwari,* RSC Advances,  2015, 5, 5311.

 6. Divergent total synthesis of 1,6,8a-tri-epi-castanospermine and 1-deoxy-6,8a-di-epi-castanospermine from       substituted azetidin-2one (β-lactam), involving a cascade sequence of reactions as key step; Dipak Kumar Tiwari, Kishor Chandra Bharadwaj, Vedavati G. Puranik  and Dharmendra Kumar Tiwari*, Org. Biomol. Chem., 2014, 12, 7389-739.

Publications from Ph.D and Post-Doc

 5. Morita–Baylis–Hillman reaction of acrylamide with isatin derivatives; R. M. Singh, K. C. Bharadwaj and Dharmendra Kumar Tiwari; Beilstein J. Org. Chem. 2014, 10, 2975-2980.

 4. Double Morita–Baylis–Hillman (MBH) strategy; an intermolecular and a chemo selective intramolecular MBH reactions for 5/6 substituted, functionalized piperidine unit. K.C. Bhardwaj and Dharmendra Kumar Tiwari, Tetrahedron, 2016, 72, 312 – 317.

 3. Enantioselective Total Synthesis of D-xylo-phytosphingosine from Substituted Azetitidin-2-one; Ganesh Pandey*, and Dharmendra Kumar Tiwari;  Tetrahedron Letters, 2009, 50, 3296-3298.

 2. Azetidin-2, 3-dione Synthon for Stereoselective Synthesis of cis and trans C-3-Alkyl/Aryl Azetidin-2-ones; Dharmendra Kumar Tiwari, A. Y. Shaikh, L. S. Pavase, V. K. Gumaste and A. R. A. S. Deshmukh. Tetrahedron, 2007, 63, 2524-2534.

 1.  Stereoselective synthesis of 3-alkylidene/alkylazetidin-2-ones from azetidin-2,3-diones; Dharmendra Kumar Tiwari,   Vikas K. Gumaste, A. R. A. S. Deshmukh;  Synthesis 2006, 01, 115-122

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